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I-Organic Intermediate CAS 158861-67-7 I-Pralmorelin Powder Ikhwalithi Engcono Kakhulu Intengo Ephansi Ikhwalithi Engcono Kakhulu Ikhwalithi Ephansi Ikhwalithi Engcono Kakhulu Intengo Ephansi

I-CAS No.158861-67-7

Ifomula C45H55N9O6

Isisindo se-Molecular 817.992

I-EINECS 206-616-8

 

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Ikhwalithi ngeke ikulahlekise futhi iphephile ngo-100%.

    Ukusetshenziswa komkhiqizo

    I-Pralmorelin (isisekelo samahhala) ivuselela ukukhiqizwa kwe-hormone yokukhula.

    ukucaciswa komkhiqizo

    Inombolo ye-CAS.
    158861-67-7
    Ifomula
    I-C45H55N9O6
    Isisindo samangqamuzana
    817.992
    Iphuzu elibilayo
    1265.3oC ku-760 mmHg
    Iphoyinti le-Flash
    719oC
    Ukuminyana
    1.27 g/cm3
    Isisindo esiqondile
    746.39000
    I-PSA  
    227.32000
    I-LogP
    5.91420
    Umfutho we-vapor
    0.0±0.3 mmHg ku-25°C
    Inkomba ye-refractive
    1.638
    Izimo zokugcina
    ?20°C
    158861-67-74qi

    Incazelo yomkhiqizo


    I-Pralmorelin, enefomula yamakhemikhali ethi C42H62N16O9, inenombolo ye-CAS 158861-67-7. Kuyi-peptide yokwenziwa esebenza njenge-analog ye-hormone-releasing hormone (GHRH). I-Pralmorelin ibonakala iyimpushana emhlophe ukuya emhlophe engenaphunga elihlukile. Isakhiwo sayo esiyisisekelo siqukethe uchungechunge lwama-amino acid axhunywe kumgogodla we-peptide. Lesi sakhi sincibilika emanzini. I-Pralmorelin ibhekwa njengephephile ukuthi isetshenziswe kuzilungiselelo zezokwelapha, kodwa ingase ibangele imiphumela engemihle efana nekhanda elibuhlungu, ukushaywa umoya, nokucanuzela kwenhliziyo. Kubalulekile ukulandela isilinganiso esifanele kanye neziqondiso zokuphatha lapho usebenzisa i-Pralmorelin.

    Izinkambu Ezisebenzayo

    Ukuntuleka Kwe-Hormone Yokukhula: I-Pralmorelin isetshenziswa ngokuyinhloko emkhakheni we-endocrinology ukuxilonga nokwelapha ukuntula kwe-hormone yokukhula. Inhloso yalo kulo mkhakha ihilela ukukhuthaza ukukhululwa kwe-hormone yokukhula kusuka ku-pituitary gland. Indlela yokusebenza yePralmorelin ihlanganisa ukubophezela kuma-receptors athile ku-hypothalamus kanye ne-pituitary gland, okuholela ekukhululweni kwe-hormone yokukhula.
    I-Muscle Mass Enhancement: I-Pralmorelin iye yafundiswa futhi ngenxa yamandla ayo okuthuthukisa imisipha namandla. Inhloso yalo kulo mkhakha ihilela ukukhuthaza ukuhlanganiswa kwamaprotheni emisipha nokunciphisa ukuwohloka kwemisipha. Indlela yokusebenza ekuthuthukisweni kwesisindo somzimba ihlanganisa ukusebenzisa i-hormone yokukhula-insulin-like growth factor 1 (IGF-1) axis, edlala indima ebalulekile ekukhuleni nasekulungiseni imisipha.


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