I-CAS 61012-19-9 I-Lecirelin enobumsulwa obuphezulu intengo ephezulu yekhwalithi ephezulu yokwaneliseka kwamakhasimende okudayiswayo okushisayo nokulethwa okusheshayo okuphephile
ukucaciswa komkhiqizo
Igama Elivamile | Lecirelin |
Inombolo ye-CAS | 61012-19-9 |
Isisindo samangqamuzana | 1209.42 |
Ukuminyana | 1.44 |
I-Molecular Formula | I-C59H84N16O12 |
IMisa ngqo | 1208.645508 |
I-PSA | 429.04000 |
Isimo sesitoreji | -20 ℃ |
Ividiyo Yomkhiqizo
Ukusetshenziswa komkhiqizo
I-Lecirelin iyi-analog yokwenziwa ye-gonadotropin-releasing hormone (GnRH). I-Lecirelin isetshenziswa kabanzi ekutadisheni ama-cysts e-ovarian follicular. Njenge-somatostatin yemvelo, i-Ranaridin iyi-peptide inhibitor yemisebenzi eminingi ye-endocrine, neuroendocrine, exocrine kanye ne-paracrine. Inobudlelwane obuhle be-peripheral somatostatin receptors (pituitary kanye ne-pancreatic), kodwa ubudlelwane obubuthakathaka be-central receptors. Lesi sici sisenza sibe nomthelela omuhle othize ekukhiqizweni kwe-hormone yokukhula kanye nokuphuma kwehomoni yokugaya ukudla. I-Ranaridin isebenza kakhulu kune-somatostatin yemvelo, futhi isikhathi sayo sokusebenza side. Umphumela wayo ovimbelayo ekukhiqizweni kwe-hormone yokukhula ukhethwa kakhulu kunalowo ekukhiqizweni kwe-insulin, okuyenza ifanelekele ukwelashwa kwe-acromegaly. Ngakolunye uhlangothi, umphumela ovimbelayo we-lanruipeptide ekukhiqizweni kwe-exocrine emathunjini, ama-hormone e-gastrointestinal kanye nendlela yokwanda kwamangqamuzana kwenza kube usizo kakhulu ekwelapheni izimila ze-endocrine emgudwini wokugaya ukudla, ikakhulukazi i-carcinoid.
Ulwazi Lwenkampani
I-Demei Pharmaceutical Technology Co., Ltd.iyibhizinisi eliguqukayo nelisungulayo elisebenza ngokukhethekile ocwaningweni, ekukhiqizeni nasekusabalaliseni izithako zokwenza imithi ezisezingeni eliphezulu nezinhlanganisela zemvelo. Ngokuzibophezela okuqinile ekuthuthukiseni imboni yezemithi yomhlaba wonke, sizinikele ekusizeni ukuthunyelwa kwemikhiqizo yezemithi yamaShayina emhlabeni wonke. Iphothifoliyo yethu yomkhiqizo ebanzi izuze ukuqashelwa ezimakethe ezibalulekile, okuhlanganisa i-UK, iJalimane, i-Australia, i-Netherlands, i-Poland, i-Russia, i-Kazakhstan, i-Philippines, i-Malaysia, i-Singapore, nezinye izifunda eziningi. Samukela izimiso zobuqotho nokungafihli lutho, sibeka kuqala ubudlelwano obuthembekile namakhasimende ethu, siqinisekisa impumelelo efanayo kanye nobudlelwano besikhathi eside.
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