I-CAS 204656-20-2 I-Liraglutide yase-China ukuthengiswa okuqondile kwefekthri okuhle kakhulu Ukuphepha Okuhlanzekile Okuphezulu ukuthunyelwa okuphezulu Ikhwalithi efanele amanani afanele ama-costomers aphezulu ukwaneliseka Ukulethwa Ngokushesha
Incazelo Yomkhiqizo
I-Liraglutide i-GLP-1(1–37) ishintshiwe kwa-Ly: iqembu le-amino lifakwe i-acylated ne-(N-hexadecanoyl)glutam- -yl moiety ebophezela ngokungaguquki kodwa ngokuzimisela ku-albumin ye-serum yomuntu. (Futhi, i-Lys ithathelwa indawo ngo-Arg.) Lezi zinguquko zihlinzeka ngeserum enwetshiwe kakhulu engu-t1?2 yamahora angu-10 kuya kwayi-15 ngemva kokuphathwa kwe-sc(0.6–1.8 mg), okuvumela ukudosa kanye ngosuku.Liraglutide (Victoza, Novo Nordisk) ilindele ukugunyazwa yi-FDA, EMEA, kanye ne-Koˉ roˉ -shoˉ (Japan).
ividiyo yomkhiqizo
Isicelo somkhiqizo
I-Liraglutide iwuhlobo olusha lomuthi we-hypoglycemic owenza kusebenze i-protein kinase ecushwe yi-AMP ngaleyo ndlela ithuthukise ukuzwela kwe-insulin. Ayigcini nje ngokuba nomphumela obalulekile we-hypoglycemic, kodwa futhi inemisebenzi yokwehlisa isisindo, ukunciphisa umfutho wegazi, kanye nokwenza ngcono iphrofayili ye-lipid yegazi.
I-Liraglutide, i-glucagon-like peptide-1 (GLP-1) receptor agonist yomuntu, yehlisa ukuphuma kwesisu, yandisa ukusutha, futhi yehlisa ukudla kwesiguli, kuyilapho inciphisa isifiso sobuchopho sokudla futhi ivumela umzimba ukuba Ukwenyuswa kwezindleko zamandla kudlala indima esisindo. ukulahlekelwa; ivimbela isibindi ekukhiqizeni i-glucose eningi futhi ikhuthaza ama-pancreas ukuthi akhiqize i-insulin eyengeziwe ukuze ehlise ushukela wegazi; ngaphezu kwalokho, i-liraglutide nayo inezinzuzo zenhliziyo nokuvikelwa kwezinso.
ukucaciswa komkhiqizo
Igama Elivamile | I-Liraglutide |
Inombolo ye-CAS | 204656-20-2 |
I-Molecular Formula | I-C172H265N43O51 |
Isisindo samangqamuzana | 3751.20000 |
I-PSA | 1513.76000 |
I-LogP | 6.12960 |
EINECS | 810-818-7 |