Ikhwalithi Engcono Kakhulu Intengo Ephansi I-CAS 148553-50-8 Pregabalin Direct Sales from China Factory Safety shipping High Purity 99% Hot Selling
Ukusetshenziswa komkhiqizo
Umuthi ungenye yezindlela zokwelapha zesithuthwane ezithembisayo kakhulu ezisathuthuka, ezisebenza kangcono kanye nokudotshwa okulula. Ingase futhi isetshenziselwe ukwelapha ubuhlungu nokukhathazeka.
ukucaciswa komkhiqizo
Inombolo ye-CAS. | 148553-50-8 |
Ifomula | I-C8H17NO2 |
Isisindo samangqamuzana | 159.22608 |
Ukuminyana | 1.0±0.1 g/cm3 |
Iphuzu elibilayo | 274.0±23.0 °C ku-760 mmHg |
Iphoyinti le-Flash | 119.5±22.6 °C |
Isisindo esiqondile | 159.125931 |
I-PSA | 63.32000 |
I-LogP | 1.12 |
Umfutho we-vapor | 0.0±1.2 mmHg ku-25°C |
Inkomba ye-refractive | 1.465 |
Izimo zokugcina | Gcina kwa-RT |
Incazelo yomkhiqizo
I-Pregabalin iyinhlanganisela yamakhemikhali ene-molecular formula C8H17NO2. Kuwumuthi owela ngaphansi kwesigaba semithi elwa nokuquleka. I-Pregabalin iphuma ku-gamma-aminobutyric acid (GABA), i-neurotransmitter ohlelweni lwezinzwa olumaphakathi. Ngokwesakhiwo, ihlobene ne-GABA ye-neurotransmitter evimbelayo, kodwa indlela yayo yokusebenza ihlukile. Ngokuya ngezakhiwo ezibonakalayo, i-pregabalin iqinile elicwebezelayo elimhlophe. Izici zayo zokuncibilika zihlanganisa ukungancibiliki emanzini kanye nokuncibilika ngokukhululekile kuzincibilikisi zemvelo ezishisayo. I-Pregabalin itholakala ngamafomu omthamo womlomo, njengamaphilisi noma amaphilisi, ukuze isetshenziswe njengomuthi.
I-Pregabalin ivame ukusetshenziselwa ukwelapha izimo ezihlukahlukene zezokwelapha, kuhlanganise nobuhlungu be-neuropathic, i-fibromyalgia, nezinhlobo ezithile zokuquleka. Isebenzisa imiphumela yayo yokwelapha ngokubophezela ku-alpha-2-delta subunit yeziteshi ze-calcium ezine-voltage-gated ohlelweni lwezinzwa olumaphakathi. Lokhu kubophezela kushintsha ukungena kwe-calcium ion, kunciphisa ukukhululwa kwama-neurotransmitters, futhi ngaleyo ndlela kunciphise ukujabula kwamangqamuzana ezinzwa.
ividiyo yomkhiqizo
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