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I-CAS 141732-76-5 Exenatide Acetate China umkhiqizi wokuthengisa oqondile inani elifanele Ikhwalithi ephezulu Ukuphepha Kokuphepha ukuhambisa okuhle kakhulu Ikhwalithi ephezulu yabathengi ukwaneliseka Ukulethwa Ngokushesha

I-peptide engu-39-amino acid ekuqaleni eyahlukanisiwe nezindlala zamathe ze-Gila monster (Heloderma suspectum), ihlukile ku-exendin-3 kuphela ezindaweni ezimbili eduze kwe-N-terminus.

 

 

 

    Incazelo Yomkhiqizo

    Ukusetshenziswa kwe-exenatide kubangela ukwanda kwe-acinar cAMP ngaphandle kokukhuthaza ukukhululwa kwe-amylase. Njenge-incretin mimetic, i-exenatide isebenza njenge-agonist ye-glucagon-like peptide-1 (GLP-1) receptor. Njenge-GLP-1, noma isebenza isikhathi eside, i-exenatide ikhulisa ukukhiqizwa kwe-insulin ngemuva kokudla futhi icindezela ukukhiqizwa kwe-glucagon. Ngenxa yalesi sizathu, i-exenatide ithole ukusetshenziswa njengomuthi wesifo sikashukela II.

    ividiyo yomkhiqizo

    Isicelo somkhiqizo

    Ukusetshenziswa kwe-exenatide acetate kubangela ukwanda kwe-acinar cAMP ngaphandle kokukhuthaza ukukhululwa kwe-amylase. Njenge-incretin mimetic, i-exenatide acetate isebenza njenge-agonist ye-glucagon-like peptide-1 (GLP-1) receptor. Njenge-GLP-1, nakuba isebenza isikhathi eside, i-exenatide acetate yandisa ukukhiqizwa kwe-insulin kwangemva kokudla futhi icindezela ukukhiqizwa kwe-glucagon. Ngalesi sizathu, i-exenatide acetate ithole ukusetshenziswa njengomuthi wesifo sikashukela II.

    ukucaciswa komkhiqizo

    Igama Elivamile Exenatide Acetate
    Inombolo ye-CAS 141732-76-5
    I-Molecular Formula
    I-C186H286N50O62S
    Isisindo samangqamuzana 4246.62000
    I-PSA  
    1812.35000
    EINECS
    1592732-453-0

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