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Dihexa CAS 1401708-83-5 Ile-iṣẹ China taara tita Sowo aabo to dara julọ Didara awọn iye owo ti o ga ni itẹlọrun Yara Ifijiṣẹ ifigagbaga idiyele giga Mimo giga

Dihexa (orukọ idagbasoke PNB-0408), ti a tun mọ ni N-hexanoic-Tyr-Ile- (6) aminohexanoic amide, jẹ oogun oligopeptide ti o wa lati angiotensin IV ti o sopọ pẹlu isunmọ giga si ifosiwewe idagbasoke hepatocyte (HGF) ati pe o ni agbara rẹ. aṣayan iṣẹ-ṣiṣe ni olugba rẹ, c-Met.

 

 

 

    ọja Apejuwe

    Pade. A ti rii agbo naa lati mu iṣẹ oye ṣiṣẹ ni agbara ni awọn awoṣe ẹranko ti ailagbara ọpọlọ-bi Alzheimer. Ninu idanwo ti iṣẹ-ṣiṣe neurotrophic, Dihexa ni a rii pe o jẹ awọn aṣẹ meje ti titobi diẹ sii ju ifosiwewe neurotrophic ti ọpọlọ ti ari.

    ọja fidio

    Ohun elo ọja

    N-Hexanoic-Gbiyanju-Ile- (6) -amino Hexanoic amide (Dihexa) jẹ angiotensin IV afọwọṣe gẹgẹbi aṣoju asọtẹlẹ / antidementia.
    Dihexa, oogun oligopeptide kan, jẹ adaṣe ẹnu ati idena ọpọlọ-ẹjẹ-permeable angiotensin IV afọwọṣe. Dihexa sopọ mọ ifosiwewe idagbasoke hepatocyte (HGF) pẹlu isunmọ giga (Kd=65 pM) ati pe o mu iṣẹ ṣiṣe rẹ pọ si ni olugba rẹ, c-Met. Dihexa ṣe afihan iṣẹ-ṣiṣe antidementia ti o dara julọ ati ilọsiwaju iṣẹ imọ ni awọn awoṣe ẹranko. Dihexa le ni agbara iwosan bi itọju aisan Alzheimer.

    ọja sipesifikesonu

    Orukọ Wọpọ Dihexa
    Nọmba CAS 1401708-83-5
    iwuwo  
    1,1 ± 0,1 g / cm3
    Ojuami farabale  
    866.2± 65.0 °C ni 760 mmHg
    Fọọmu Molecular
    C27H44N4O5
    Òṣuwọn Molikula 504.662
    LogP  
    2.78
    EINECS
    227-005-2
    Oru Ipa  
    0.0±0.3 mmHg ni 25°C
    Atọka ti Refraction
    1.529

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