Umgangatho oPhezulu wokuThengisa ngokuthe ngqo kwiFactory yaseChina CAS 736992-21-5 Elamipretide enexabiso elinomtsalane kwintengiso eshushu isitokhwe kunye nokhuseleko lwamasiko kwindlu ngendlu
ukucaciswa kwemveliso
Igama eliqhelekileyo | Iiprets ezihlalayo |
Inombolo yeCAS | 736992-21-5 |
Ubunzima beMolekyuli | 639.79 |
Ifomula yeemolekyuli | C32H49N9O5 |
EINECS | 205-858-1 |
Ukuxinana | 1.34±0.1 g/cm3(Kuxelwe kwangaphambili) |
Indawo yokubilisa | N / A |
Uzinzo | Hygroscopic |
IMisa ngqo | 639.38600 |
PSA | 276.02000 |
Imeko yokugcina | -20°C |
Ividiyo yeMveliso
Ukusetyenziswa kweMveliso
I-Elamipretide (MTP-131, SS-31, D-Arg-DMT-Ls-PHE-NH2) yi-inhibitor ye-cytochrome c peroxidase. I-Elamipretide inokuphucula ukungasebenzi kakuhle kwe-mitochondrial, i-synapse kunye nokuphazamiseka kwememori okubangelwa yi-lipopolysaccharide kwiimpuku.
I-elamipretide acetate yi-molecule encinci ye-polypeptide eyenziwe ngee-amino acids ezine. Kwi-vivo, ijolise kwi-membrane yangaphakathi ye-mitochondria, enokuthintela iiseli ze-nerve kunye nezinye iintlobo zeeseli kwi-oxidative Chemicalbook umonakalo. Thintela i-mitochondrial depolarization, ukunciphisa i-islet cell apoptosis, ukwandisa isivuno se-islet cell kunye nokuphucula umsebenzi emva kokutshintshwa. Iziyobisi ezine-Elamipretide acetate njengezona zinto ziphambili zingena kwisigaba sesithathu seklinikhi.
Ulwazi lweNkampani
I-Demei Pharmaceutical Technology Co., Ltd.lishishini eliguquguqukayo neliyintshayo eligxile kuphando, ukuvelisa, kunye nokusasazwa kwezithako zamayeza ezikumgangatho ophezulu kunye neekhompawundi eziphilayo. Ngokuzibophelela ngokuqinileyo ekuqhubeleni phambili ishishini loxubo mayeza lehlabathi, sizinikele ekuququzeleleni ukuthunyelwa kwemveliso yamayeza eTshayina kwihlabathi liphela. Ipotfoliyo yethu yemveliso ebanzi iye yafumana ukuqondwa kwiimarike eziphambili, kuquka i-UK, iJamani, i-Australia, iNetherlands, iPoland, iRashiya, iKazakhstan, iiPhilippines, iMalaysia, iSingapore, kunye neminye imimandla emininzi. Ukwamkela imigaqo yemfezeko kunye nokungafihli, sibeka phambili ukwakha ubudlelwane obuthembekileyo kunye nabathengi bethu, siqinisekisa impumelelo efanayo kunye nobudlelwane bexesha elide.
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