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I-Tetracaine CAS 94-24-6 5094-24-6 iNtengiso ngokuthe ngqo evela e-China Ukuhlambuluka okuPhakamileyo kweXabiso eliPhantsi loKhuseleko ukuhanjiswa ngokukhawuleza

I-Tetracaine sisithomalalisi se-topical yendawo yamehlo; isebenza ngokuphazamisa ukungena kwee-ion zesodium kwiiseli zemithambo-luvo.

    Ingcaciso yeMveliso

    I-Tetracaine liyeza lendawo lokuthomalalisa iintlungu okanye leyeza lokuthomalalisa umqala, amehlo, okanye impumlo. Ngokuqhelekileyo, ichiza lilawulwa phambi kokuba uqalise utyando ukunciphisa intlungu kwinkqubo. I-Tetracaine isetyenziswe emehlweni imizuzu engama-30 ngaphambi kokuqala kwe-intravenous kunye nemiphumo yayo ingahlala ukuya kwimizuzu eyi-15.

    ividiyo yemveliso

    Isicelo seMveliso

    I-Tetracaine isetyenziselwa ukuvavanya amandla okusebenzisana kweziyobisi-nanoparticle ukuze kuphuculwe ukungena kweziyobisi esikhumbeni.
    I-Tetracaine topical (yesikhumba) isetyenziselwa ukuba ndindisholo amalungu ahlukeneyo omzimba phambi kwenkqubo yotyando okanye uvavanyo lwezonyango. Ngokuchaseneyo, i-tetracaine ophthalmic drops isetyenziswa njenge-anesthetic yendawo yamehlo.
    I-Tetracaine isetyenziswe njenge-anesthetic kunye nokunciphisa i-glucose synthesis kwi-infusions yamathumbu amancinci amancinci. Kwakhona kusetyenziswe ukuvimbela i-ryanodine receptors (RyRs) kwiigundane.
    I-Tetracaine isetyenziswe njenge-anesthetic kunye nokunciphisa i-glucose synthesis kwi-infusions yamathumbu amancinci amancinci. Kwakhona kusetyenziswe ukuvimbela i-ryanodine receptors (RyRs) kwiigundane.
    I-Tetracaine hydrochloride (i-Pontocaine) yi-ester ye-PABA eyi-ejenti esebenzayo ye-anesthetic yendawo kwaye iqhele ukusetyenziswa kwi-spinal (subarachnoid) i-anesthesia. I-epinephrine yongezwa rhoqo ukwandisa ixesha le-anesthesia. ITetracaine inamandla kakhulu kwaye inetyhefu ngakumbi kuneprocaine kunye necocaine. Inokuqala kwemizuzu emi-5 kunye neeyure ezi-2 ukuya kwezi-3 zesenzo.

    ukucaciswa kwemveliso

    Ukuxinana 1.0±0.1 g/cm³
    Indawo yokubilisa 389.4±27.0 °C kwi-760 mmHg
    Indawo yokunyibilika 43 °C
    Ifomula yeemolekyuli I-C15H24N2O2
    Ubunzima beMolekyuli 264.363
    Indawo yokuflasha 189.3±23.7 °C
    IMisa ngqo 264.183777
    PSA 41.57000
    LogP 3.65
    Uxinzelelo lomphunga 0.0±0.9 mmHg ku-25°C
    Isalathiso seRefraction 1.538
    Imbonakalo Umgubo omhlophe

    Iphakheji

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