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I-Procaine CAS 59-46-1 Umgangatho ogqwesileyo oBonelekileyo obuBonelekileyo obuBonelekileyo Umgangatho oPhezulu oPhezulu oPhezulu wexabiso eliPhezulu.

Inendima njengeyeza lendawo yokuthomalalisa iintlungu, i-central nervous system depressant, ichiza le-peripheral nervous system kunye ne-allergen yeziyobisi.

    Ingcaciso yeMveliso

    Inendima njengeyeza lendawo yokuthomalalisa iintlungu, i-central nervous system depressant, ichiza le-peripheral nervous system kunye ne-allergen yeziyobisi.
    Indlela esisiseko ye-analgesia ephantsi kwayo yonke i-anesthetics yendawo kukuthintelwa kwe-neurotransmission ngokuthintelwa kweziteshi ze-sodium kunye ne-nerve fibers. Iprocaine isebenza ikakhulu ngokuthintela ukungena kwesodium ngevolthi gated iziteshi zesodium kwi-neuronal cell membrane ye-peripheral nerves. Xa ukungena kwe-sodium kuphazamiseka, isenzo esinokuthi singakwazi ukuvela kwaye ukuqhutyelwa kwesignali kunqatshelwe.
    I-Procaine (i-Novocain) isetyenziswa kakhulu kwiinkqubo zamazinyo okanye zonyango ezifuna i-anesthesia yokungena, i-peripheral block, okanye i-spinal block.

    ividiyo yemveliso

    Isicelo seMveliso

    Iprocaine ikhawuleza kakhulu imetaboliseni kwiplasma ngecholinesterases nakwisibindi nge-ester hydrolysis ngepseudocholinesterase. Ubomi besiqingatha se-in vitroelimination bumalunga nemizuzwana engama-60. Nayiphi na imeko enciphisa ugxininiso lwe-cholinesterase inokunyusa ukuvezwa kwiprocaine kunye netyhefu enokubakho. Ukuncipha komsebenzi we-enzyme kunokufunyanwa ngokusilela kwemfuza, isifo sesibindi, isifo esibi, ukungondleki, ukusilela kwezintso, ukutshisa, i-thirdtrimester yokukhulelwa, kunye nokulandela utyando lwe-cardiopulmonary bypasssurgery. I-Ester hydrolysis ivelisa i-PABA, i-compounds enoxanduva lokwaliwa okuxhaphakileyo kwi-ester anesthetics. Iprocaine ayisetyenziswanga ngokwesihloko ngenxa yokungakwazi ukudlula kwi-lipid membranes kwaye ifumana ukusetyenziswa njenge-aninfiltration agent ye-cutaneous okanye i-mucous membranes, iinkqubo ezimfutshane. Iprocaine ikwasetyenziselwa i-peripheral nerveblock kunye ne-epidural agent ukuxilonga ii-syndromes zentlungu.

    ukucaciswa kwemveliso

    Ukuxinana 1.1±0.1 g/cm3
    Indawo yokubilisa 373.6±22.0 °C kwi-760 mmHg
    Indawo yokunyibilika 61oC
    Ifomula yeemolekyuli I-C13H20N2O2
    Ubunzima beMolekyuli 236.310
    Indawo yokuflasha 179.8±22.3 °C
    IMisa ngqo 236.152481
    PSA 55.56000
    LogP 2.36
    Uxinzelelo lomphunga 0.0±0.8 mmHg ku-25°C
    Isalathiso seRefraction 1.543
    Imbonakalo Okumhlophe Okuqinileyo

    Iphakheji

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    Iimveliso zexabiso eliphezulu kunye nendalo ye-R&D Ithunyelwe kwiibhotile ezine-fluorinated

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    Umthumeli wempahla uya kukhupha inombolo yokulandelela kumazwe ngamazwe ngosuku okanye ngosuku olulandelayo lokufika.
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    Umzi-mveliso wethu unemveliso yonyaka ezinzileyo yeetoni ezingama-50,000 zemathiriyeli ekrwada unyaka wonke. Ikhonkco lemveliso kunye nekhonkco lokuthengisa liyaqhubeka nokuhlutha. Indawo yethu yokugcina inomthamo omkhulu womgubo kunye nesitokhwe solwelo. Siyabamkela abantu abavela kuzo zonke iinkalo zobomi ukuba baxhase kwaye basebenzisane.
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