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Ubonelelo loMvelisi ngezinto ezikrwada CAS 113-79-1 Argipressin Umgangatho oMgangatho oLona xabiso liphantsi ukuHanjiswa ngokuKhawuleza uKhuseleko ngenqanawe ukuPhucuka okuphezulu 99%

Inombolo yeCAS 113-79-1

Ifomula yeC46H65N15O12S2

Ubunzima beMolekyuli 1084.2316

I-EINECS 204-035-4

 

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Umgangatho awuyi kukuvumela ukuba uphantsi kwaye i-100% ikhuselekile

    Ukusetyenziswa kwemveliso

    I-Argipressin ibophelela kwi-arginine vasopressin receptor V1 ene-Kd ye-1.31 nM kwiiseli ze-A7r5 zegundane ze-aortic ezigudileyo.

    ukucaciswa kwemveliso

    Inombolo yeCAS.
    113-79-1
    Ifomula
    I-C46H65N15O12S2
    Ubunzima bemolekyuli
    1084.2316
    Ukuxinana
    1.6±0.1 g/cm3
    Indawo yokuflasha
    113℃
    Ubunzima obuchanekileyo
    1083.437866
    PSA  
    512.03000
    LogP
    -5.99
    Imbonakalo
    umgubo omhlophe
    Isalathiso sokuqhafaza
    1.724
    Iimeko zokugcina
    2-8°C
    113-79-1w2n

    Ingcaciso yeMveliso


    I-ChEBI: Eyona ndlela iphambili ye-mammalian vasopressin (ihomoni ye-antidiuretic). I-nonapeptide equkethe i-arginine kwi-residue ye-8 kunye ne-cysteines ezimbini ze-disulfide-linked kwi-residus ye-1 kunye ne-6. I-Vasopressin tannate (i-PitressinTannate) yi-tannate engenamanzi e-vasopressin elawulwa nge-intramuscularly (1.5-5.0 ye-pressor ye-unit long ye-protectors) isenzo ngokukhutshwa kancinci kwevasopressin.


    Imimandla Esebenzayo

    IArgipressin lolona hlobo lubalaseleyo lwemammalian vasopressin (ihomoni ye-antidiuretic). I-nonapeptide equkethe i-arginine kwi-residue ye-8 kunye ne-cysteines ezimbini ze-disulfide-linked kwi-residus ye-1 kunye ne-6. Inendima njengeziyobisi ze-cardiovascular, i-hematologic agent kunye ne-mitogen.|Impembelelo ye-physiologic ye-vasopressin yindlela ye-Vasoconstriction , kunye nokuncipha kweDiuresis.|Argipressin yipeptide yokwenziwa efana ne-endogenous nonapeptide hormone enepropathi ye-antidiuretic. Ihlanganiswe kwi-hypothalamus kwaye igcinwe / ikhutshwe kwi-lobe yangasemva ye-pituitary, umsebenzi oyintloko we-argipressin ulawula umthamo we-extracellular fluid. Le arhente inokusebenza njenge-vasoconstrictor, inyusa uxinzelelo lwegazi kunye ne-systemic vascular resistance.|Olona hlobo luphambili lwehomoni ye-mammalian antidiuretic. I-nonapeptide equkethe i-ARGININE kwi-residue ye-8 kunye ne-cysteines ezimbini ze-disulfide-linked kwi-residues ze-1 kunye ne-6. I-Arg-vasopressin isetyenziselwa ukunyanga i-DIABETES INSIPIDUS okanye ukuphucula ithoni ye-vasomotor kunye noxinzelelo lwegazi.

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