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Umenzi wePowder ephezulu 98% yePeptides Powder Liraglutide CAS 204656-20-2 Peptides Powder kwiVials ngexabiso eliphantsi ubuhle bepeptides Izinto zokuthambisa

Igama lemveliso: Liraglutide

Inombolo yeCAS: 204656-20-2

Ifomula yemolekyuli:C172H265N43O51

Ubunzima bemolekyuli:3751.202

I-EINECS No.: 810-818-7

 

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    ukucaciswa kwemveliso

    Igama lemveliso ILiraglutide
    Inombolo yeCAS. 204656-20-2
    I-EINECS No. 810-818-7
    Ukuxinana N / A
    Indawo yokubilisa N / A
    Indawo yokunyibilika N / A
    Indawo yokuflasha N / A
    Ifomula yemolekyuli C172H265N43O51
    Ubunzima bemolekyuli 3751.202
    Imbonakalo Umgubo oMhlophe
    Iimeko zokugcina -20°C

    ividiyo yemveliso

    Ingcaciso yeMveliso

    I-Liraglutide (NN2211) yi-glucagon-efana ne-peptide-1 receptor agonist yexesha elide. Ithengiswa phantsi kwegama le-brand Victoza, lichiza elitofwayo eliphuhliswe nguNovo Nordisk kunyango lwe-2 yeswekile. Ngo-2015, i-Novo Nordisk yaqala ukuyithengisa e-US phantsi kwegama le-brand liraglutide njengonyango lokutyeba kubantu abadala ubuncinci ubuncinci bemeko ye-comorbid enxulumene nobunzima.
    Usetyenziso lwezonyango
    ILiraglutide sisitofu esiphuma kanye yonke imihla se-incretin yomntu (ihomoni ye-metabolic) iglucagon-efana ne-peptide-1 (GLP-1), kunyango lwe-2 yeswekile okanye ukutyeba.
    Uhlobo lwesi-2 seswekile
    ILiraglutide iphucula ulawulo lweswekile yegazi. Ukulibazisa ukukhupha isisu, kunye nokucinezela i-prandial glucagon secretion.
    Ngokuqhelekileyo kwiidigri ezahlukeneyo kunye nezinye i-GLP-1 receptor agonists, i-liraglutide ineengenelo kunyango lwemveli lohlobo lwesi-2 seswekile:
    Inamandla okuthintela i-apoptosis kunye nokuvuselela ukuvuselelwa kweeseli ze-beta (ezibonwa kwizifundo zezilwanyana).
    Yehlisa umdla wokutya kwaye inqande ukufumana ubunzima bomzimba, njengoko kubonisiwe kuphononongo lwentloko ukuya entloko ngokuchasene ne-glimepiride.
    Yehlisa amanqanaba e-triglyceride yegazi.
    Ukutyeba ngokugqithiseleyo
    I-Liraglutide yamkelwe njengesixhobo esitofwayo kukutya okunekhalori encitshisiweyo kunye nokwandisa umsebenzi womzimba wolawulo lobunzima obungapheliyo kwizigulana zabantu abadala. Iikhrayitheriya ezikhankanyiweyo ziinkomba zobunzima bomzimba wokuqala (BMI) we-30 kg/m2 okanye ngaphezulu (okutyebileyo), okanye i-27 kg/m2 okanye ngaphezulu (ubunzima obugqithisileyo), phambi kokuba ubuncinci bube bubunzima obunxulumene nemeko ye-comorbid (umzekelo, uxinzelelo lwegazi, uhlobo lwe-2 yesifo sikashukela, okanye i-dyslipidemia). Ngasekupheleni kwe-2014, idatha yaxelwa kwi-SCALE ™ Ukutyeba kakhulu kunye nolingo lwe-Prediabetes, oluyi-randomized, i-double-blind, i-placebo-controlled, uvavanyo lwezizwe ngezizwe kubantu abangenasifo seswekile kunye nokukhuluphala kunye nabantu abangenasifo seswekile abanobunzima kunye ne-comorbidities. Kwesi sigaba sesi-3 solingo, bekukho abathathi-nxaxheba be-3,731 abangabalulekanga kunyango nge-liraglutide 3 mg okanye i-placebo, zombini ngokudityaniswa nokutya kunye nokuzilolonga. Abo bagqibe uvavanyo lweeveki ezingama-56 bafumana ukwehla kobunzima obuphakathi kwe-9.2%, xa kuthelekiswa nokuncipha kwe-3.5% kwiqela le-placebo.

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