Kushushu ukuthengisa umgangatho ophezulu 98% Polypeptide Leuprorelin acetate powder CAS 74381-53-6 evela kumthengisi waseTshayina ngexabiso eliphantsi Ukuhanjiswa okuKhuselekileyo
ukucaciswa kwemveliso
Igama lemveliso | Leuprorelin acetate |
Inombolo yeCAS. | 74381-53-6 |
I-EINECS No. | 686-285-8 |
Ukuxinana | N / A |
Indawo yokubilisa | 1720.5ºC ku-760 mmHg |
Indawo yokunyibilika | 150-155ºC |
Indawo yokuflasha | 994.3ºC |
Ifomula yemolekyuli | I-C61H88N16O14 |
Ubunzima bemolekyuli | 1269.47 |
Imbonakalo | Umgubo oMhlophe |
Iimeko zokugcina | -20°C |
ividiyo yemveliso
Ingcaciso yeMveliso
I-Leuprorelin acetate, kunye ne-chemical formula C59H84N16O12, inenombolo ye-CAS 74381-53-6. Yi-analog ye-peptide yokwenziwa ye-gonadotropin-releasing hormone (GnRH). I-Leuprorelin acetate ibonakala njengomgubo omhlophe ukuya kumhlophe ngaphandle kwevumba elahlukileyo. Isakhiwo sayo esisisiseko siquka ikhonkco le-peptide kunye ne-amino acids eqhotyoshelwe kwiqela le-acetate. Le khompawundi iyanyibilika emanzini. I-Leuprorelin acetate ithathwa njengento ekhuselekileyo yokusetyenziswa kwizicelo zonyango.
Imimandla Esebenzayo
Unyango lweCancer: I-Leuprorelin acetate isetyenziswa ngokuqhelekileyo kunyango lwee-cancer ezixhomekeke kwi-hormone ezifana nomdlavuza we-prostate kunye nomhlaza webele. Indlela yayo yokusebenza kunyango lomhlaza ibandakanya ukucinezelwa kwehomoni ekhupha i-gonadotropin (GnRH), ekhokelela ekunciphiseni ukuveliswa kweehomoni zesini ezifana ne-testosterone kunye ne-estrogen. Olu xinzelelo lwehomoni lunokunceda ukucothisa ukukhula kwamathumba axhomekeke kwihomoni.
I-Endometriosis: I-Leuprorelin acetate ikwasetyenziswa kunyango lwe-endometriosis, imeko apho ithishu ehlala esibelekweni ikhule ngaphandle kwayo. Kulo mongo, indlela yokusebenza iyafana nokusetyenziswa kwayo kunyango lomhlaza, apho icinezela ukuveliswa kweehomoni zesini kwaye inceda ukunciphisa iimpawu ezinxulumene ne-endometriosis.
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