Intengiso eshushu iStokhwe esiLungileyo iXabiso eliLihle le-CAS 204656-20-2 iLiraglutide iThengisa ngokuThengisa ngokuthe ngqo kwiFactory yaseChina ngokuthumela ngenqanawa
Ukusetyenziswa kwemveliso
I-Liraglutide yi-glucagon-like peptide-1 (GLP-1) i-receptor agonist esetyenziselwa ukunyanga isifo seswekile se-2.
ukucaciswa kwemveliso
Inombolo yeCAS. | 204656-20-2 |
Ifomula | C172H265N43O51 |
Ubunzima bemolekyuli | 3751.262 |
Ubunzima obuchanekileyo | 3748.95000 |
PSA | 1513.76000 |
LogP | 6.12960 |
Iimeko zokugcina | -20°C |
Ingcaciso yeMveliso
I-Liraglutide, kunye ne-chemical formula C172H265N43O51, inenombolo ye-CAS 204656-20-2. Yihomoni ye-peptide yeklasi ye-glucagon-like peptide-1 (GLP-1) receptor agonists. ILiraglutide ibonakala ingenambala ukuya kulwelo olutyheli kancinci kwaye akukho vumba lahlukileyo. Isakhiwo sayo esisisiseko siquka ikhonkco elide le-amino acids. Le khompawundi iyanyibilika emanzini. ILiraglutide ithathwa njengekhuselekile ukuba isetyenziswe kunyango lweswekile kunye nokutyeba. Nangona kunjalo, kunokubangela iziphumo ebezingalindelekanga ezifana nesicaphucaphu, ukuhlanza, kunye norhudo. Kubalulekile ukulandela idosi emiselweyo kwaye udibane nochwepheshe bezempilo ukuze usetyenziswe ngokufanelekileyo. ILiraglutide kufuneka igcinwe kwindawo epholileyo neyomileyo, kude nelanga elithe ngqo.
Imimandla Esebenzayo
Unyango lweswekile: ILiraglutide isetyenziswa ikakhulu kunyango lwesifo seswekile esi-2. Isebenza ngokuvuselela ukukhutshwa kwe-insulin kunye nokunciphisa ukuveliswa kweglucagon, okukhokelela ekunciphiseni amanqanaba eswekile yegazi. Indlela yokusebenza ibandakanya ukubophelela kwi-GLP-1 receptors kwi-pancreas, ephucula ukukhuselwa kwe-insulin exhomekeke kwiglucose kwaye ikhuthaze ukuhlutha.
Ulawulo lobunzima: ILiraglutide ikwavunyiwe kunyango lokutyeba kakhulu. Inceda ekulawuleni ubunzima ngokunciphisa umdla wokutya kunye nokukhuthaza ukuziva ugcwele. Indlela yokusebenza kulo mongo iyafana nefuthe layo kwisifo seswekile, njengoko isebenza kwi-GLP-1 receptors ukulawula ukutya kunye nokulinganisela kwamandla.
ividiyo yemveliso
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