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Umvelisi waseTshayina unikezela nge-98% ukucoceka okuphezulu kwe-Rosiptor powder kunye nexabiso elihle CAS 782487-28-9 Ukhuseleko lweCustoms Ukuhanjiswa ngokukhawuleza

Igama lemveliso: Rosiptor

Inombolo yeCAS: 782487-28-9

Ifomula yemolekyuli:C20H35NO2

Ubunzima bemolekyuli:321.5

I-EINECS No.: 200-001-8

 

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    ukucaciswa kwemveliso

    Igama lemveliso Rosiptor
    Inombolo yeCAS. 782487-28-9
    I-EINECS No. 200-001-8
    Ukuxinana 1.1±0.1 g/cm3
    Indawo yokubilisa 451.6±45.0 °C(Kuqikelelwe)
    Indawo yokunyibilika N / A
    Indawo yokuflasha 226.9±28.7 °C
    Ifomula yemolekyuli C20H35NO2
    Ubunzima bemolekyuli 321.5
    Imbonakalo Umgubo oMhlophe
    Iimeko zokugcina -20°C

    ividiyo yemveliso

    Ingcaciso yeMveliso:

    I-Retatrutide yi-molecule yophando eyenza i-receptors yomzimba isebenze kwiihomoni ezintathu - iglucagon, i-insulinotropic polypeptide exhomekeke kwi-glucose (GIP), kunye ne-glucagon-like peptide-1 (GLP-1), kwaye ifundelwa unyango lokutyeba.
    Isebenzisa i-triple-agonist (i-triple-G) indlela yokwenza. Ukongeza ekubeni yi-GLP-1RA, ikwajolise kwi-gastric inhibitory polypeptide receptor (GIPR), kunye ne-glucagon receptor (GCGR). Oku ngenxa yoko kubonise iinzuzo ezongeziweyo ezisebenzayo kwiimvavanyo zeklinikhi, eziphakamileyo kunezo zibonwa nge-W, eziququzelela malunga ne-15% yokulahlekelwa kwesisindo somzimba.
    I-Semaglutide i-polypeptide equlethe ukulandelelana komgca we-31 amino acids ehlanganiswe kunye ne-peptide linkages. I-agonist ye-glucagon-like peptide 1 receptors (GLP1 AR) kwaye isetyenziselwa unyango lwe-2 yeswekile.
    Inendima njenge-agent ye-hypoglycemic, i-glucagon-like peptide-1 receptor agonist, i-anti-obesity agent, i-neuroprotective agent kunye ne-appetite depressant. Yipolypeptide kunye ne-lipopeptide.

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