Umvelisi waseTshayina unikezela nge-98% ukucoceka okuphezulu kwe-Rosiptor powder kunye nexabiso elihle CAS 782487-28-9 Ukhuseleko lweCustoms Ukuhanjiswa ngokukhawuleza
ukucaciswa kwemveliso
Igama lemveliso | Rosiptor |
Inombolo yeCAS. | 782487-28-9 |
I-EINECS No. | 200-001-8 |
Ukuxinana | 1.1±0.1 g/cm3 |
Indawo yokubilisa | 451.6±45.0 °C(Kuqikelelwe) |
Indawo yokunyibilika | N / A |
Indawo yokuflasha | 226.9±28.7 °C |
Ifomula yemolekyuli | C20H35NO2 |
Ubunzima bemolekyuli | 321.5 |
Imbonakalo | Umgubo oMhlophe |
Iimeko zokugcina | -20°C |
ividiyo yemveliso
Ingcaciso yeMveliso:
I-Retatrutide yi-molecule yophando eyenza i-receptors yomzimba isebenze kwiihomoni ezintathu - iglucagon, i-insulinotropic polypeptide exhomekeke kwi-glucose (GIP), kunye ne-glucagon-like peptide-1 (GLP-1), kwaye ifundelwa unyango lokutyeba.
Isebenzisa i-triple-agonist (i-triple-G) indlela yokwenza. Ukongeza ekubeni yi-GLP-1RA, ikwajolise kwi-gastric inhibitory polypeptide receptor (GIPR), kunye ne-glucagon receptor (GCGR). Oku ngenxa yoko kubonise iinzuzo ezongeziweyo ezisebenzayo kwiimvavanyo zeklinikhi, eziphakamileyo kunezo zibonwa nge-W, eziququzelela malunga ne-15% yokulahlekelwa kwesisindo somzimba.
I-Semaglutide i-polypeptide equlethe ukulandelelana komgca we-31 amino acids ehlanganiswe kunye ne-peptide linkages. I-agonist ye-glucagon-like peptide 1 receptors (GLP1 AR) kwaye isetyenziselwa unyango lwe-2 yeswekile.
Inendima njenge-agent ye-hypoglycemic, i-glucagon-like peptide-1 receptor agonist, i-anti-obesity agent, i-neuroprotective agent kunye ne-appetite depressant. Yipolypeptide kunye ne-lipopeptide.
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