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I-CAS 170851-70-4 Ifektri yase-Ipamorelin yaseChina ibonelela ngomgangatho olungileyo kunye nokusulungeka okuphezulu kwexabiso eliphantsi kunye nokwaneliseka okuphezulu kwabathengi ngokukhawuleza ukuhanjiswa okukhuselekileyo.

I-Ipamorelin (INN) (igama lekhowudi yokuphuhlisa i-NNC 26-0161) i-agonist ekhethiweyo ye-peptide ye-ghrelin / i-hormone yokukhula secretagogue receptor (GHS) kunye ne-hormone yokukhula secretagogue. I-2-Nal-D-Phe-Lys-NH2 eyayithathwe kwi-GHRP-1.

 

 

    Ingcaciso yeMveliso

    I-Ipamorelin (INN) (igama lekhowudi yophuhliso i-NNC 26-0161) i-agonist ekhethiweyo ye-peptide ye-ghrelin / i-hormone yokukhula secretagogue receptor (GHS) kunye ne-hormone yokukhula secretagogue. I-2-Nal-D-Phe-Lys-NH2 eyayithathwe kwi-GHRP-1.

    ividiyo yemveliso

    Isicelo seMveliso

    I-Ipamorelin ekuqaleni yaphuhliswa nguNovo Nordisk, kwaye yaphandwa kwizilingo zekliniki zesigaba II yi-Helsinn Therapeutics yonyango lwe-ileus yangemva kokusebenza, kodwa yayekwa ngenxa yokungabikho kokusebenza kakuhle.I-Ipamorelin isetyenziswe ngabadlali njengeyeza lokuphucula ukusebenza.

    ukucaciswa kwemveliso

    Igama eliqhelekileyo Ipamorelin
    Inombolo yeCAS 170851-70-4
    Ukuxinana  
    1.3±0.1 g/cm3
    Indawo yokubilisa  
     1185.5±65.0 °C kwi-760 mmHg
    Ifomula yeemolekyuli
    C38H49N9O5
    Ubunzima beMolekyuli 711.853
    PSA  
    240.21000
    LogP  
    1.72
    EINECS
    227-005-2
    Uxinzelelo lomphunga  
    0.0±0.3 mmHg ku-25°C
    Isalathiso seRefraction
    1.624

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