I-CAS 170851-70-4 Ifektri yase-Ipamorelin yaseChina ibonelela ngomgangatho olungileyo kunye nokusulungeka okuphezulu kwexabiso eliphantsi kunye nokwaneliseka okuphezulu kwabathengi ngokukhawuleza ukuhanjiswa okukhuselekileyo.
Ingcaciso yeMveliso
I-Ipamorelin (INN) (igama lekhowudi yophuhliso i-NNC 26-0161) i-agonist ekhethiweyo ye-peptide ye-ghrelin / i-hormone yokukhula secretagogue receptor (GHS) kunye ne-hormone yokukhula secretagogue. I-2-Nal-D-Phe-Lys-NH2 eyayithathwe kwi-GHRP-1.
ividiyo yemveliso
Isicelo seMveliso
I-Ipamorelin ekuqaleni yaphuhliswa nguNovo Nordisk, kwaye yaphandwa kwizilingo zekliniki zesigaba II yi-Helsinn Therapeutics yonyango lwe-ileus yangemva kokusebenza, kodwa yayekwa ngenxa yokungabikho kokusebenza kakuhle.I-Ipamorelin isetyenziswe ngabadlali njengeyeza lokuphucula ukusebenza.
ukucaciswa kwemveliso
Igama eliqhelekileyo | Ipamorelin |
Inombolo yeCAS | 170851-70-4 |
Ukuxinana | 1.3±0.1 g/cm3 |
Indawo yokubilisa | 1185.5±65.0 °C kwi-760 mmHg |
Ifomula yeemolekyuli | C38H49N9O5 |
Ubunzima beMolekyuli | 711.853 |
PSA | 240.21000 |
LogP | 1.72 |
EINECS | 227-005-2 |
Uxinzelelo lomphunga | 0.0±0.3 mmHg ku-25°C |
Isalathiso seRefraction | 1.624 |