Umgangatho oPhezulu oPhantsi ngexabiso eliphantsi CAS 148553-50-8 Pregabalin Ukuthengiswa ngokuthe ngqo ukusuka kwiFactory yaseChina ukuhambisa uKhuseleko oluPhezulu 99% Ukuthengisa okushushu
Ukusetyenziswa kwemveliso
Ichiza lolona nyango luthembisayo lokuxhuzula kuphuhliso, olusebenza ngcono kunye nokudosa lula. Ingasetyenziselwa ukunyanga iintlungu kunye nokuxhalaba.
ukucaciswa kwemveliso
Inombolo yeCAS. | 148553-50-8 |
Ifomula | C8H17NO2 |
Ubunzima bemolekyuli | 159.22608 |
Ukuxinana | 1.0±0.1 g/cm3 |
Indawo yokubilisa | 274.0±23.0 °C kwi-760 mmHg |
Indawo yokuflasha | 119.5±22.6 °C |
Ubunzima obuchanekileyo | 159.125931 |
PSA | 63.32000 |
LogP | 1.12 |
Uxinzelelo lomphunga | 0.0±1.2 mmHg ku-25°C |
Isalathiso sokuqhafaza | 1.465 |
Iimeko zokugcina | Gcina eRT |
Ingcaciso yeMveliso
I-Pregabalin yi-chemical compound kunye ne-molecular formula C8H17NO2. Liyeza eliwela phantsi kweklasi yamachiza e-anticonvulsant. I-Pregabalin yi-derivative ye-gamma-aminobutyric acid (GABA), i-neurotransmitter kwinkqubo ye-nervous central. Ngokwesakhiwo, inxulumene ne-GABA ye-neurotransmitter ye-inhibitory, kodwa indlela yokusebenza kwayo yahlukile. Ngokubhekiselele kwiipropati zomzimba, i-pregabalin yikristale emhlophe eqinileyo. Iimpawu zayo zokunyibilika zibandakanya ukunganyibiliki ngokoqobo emanzini kunye nokunyibilika ngokukhululekileyo kwizinyibilikisi zendalo ezikwipolar. I-Pregabalin ifumaneka kwiifom zedosi yomlomo, njengee-capsules okanye iipilisi, ukusetyenziswa kweyeza.
I-Pregabalin isetyenziswa ngokuqhelekileyo ukunyanga iimeko ezahlukeneyo zonyango, kubandakanywa intlungu ye-neuropathic, i-fibromyalgia, kunye neentlobo ezithile zokubamba. Isebenzisa iziphumo zayo zonyango ngokuzibophelela kwi-alpha-2-delta subunit ye-voltage-gated calcium channels kwinkqubo ye-nervous central. Oku kubopha kumodareyitha ukungena kwe-calcium ion, ukunciphisa ukukhululwa kwee-neurotransmitters, kwaye ngaloo ndlela kunciphisa ukonwaba kweeseli zemithambo-luvo.
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Umgubo: ingxowa yefoyile ephindwe kabini yealuminiyam yesampulu eyi-1kg, kunye ne-25kgs ngegubu ngalinye ngobuninzi
Ulwelo: ibhotile etywiniweyo kwisampulu ye-1L, kunye ne-25kgs ngegubu ngalinye ngobuninzi