Ukuthengiswa ngokuthe ngqo kwi-China Factory CAS 1006376-62-0(1R,2R)-2-(3,4-difluorophenyl)cyclopropane carboxaMide Hot Sale Stock
ukucaciswa kwemveliso
Inombolo yeCAS. | 1006376-62-0 |
Ifomula | C10H9F2NO |
Ubunzima bemolekyuli | 197.181 |
Ukuxinana | 1.4±0.1 g/cm3 |
Indawo yokubilisa | 347.9±42.0 °C kwi-760 mmHg |
Indawo yokuflasha | 164.2±27.9 °C |
Ubunzima obuchanekileyo | 197.065216 |
PSA | 44.08000 |
LogP | 0.65 |
Uxinzelelo lomphunga | 0.0±0.8 mmHg ku-25°C |
Isalathiso sokuqhafaza | 1.556 |
Ingcaciso yeMveliso
I-Ticagrelor sisiyobisi se-antiplatelet yomlomo, igama layo le-brand brand yaseMelika nguBrilinta, kunye negama layo laseYurophu yiBrilique. I-Ticagrelor i-reversible platelet adenosine diphosphate (ADP) i-receptor antagonist eyenzelwe ukuthintela iiplatelet ukuba zibambene kunye nokwenza amacwecwe egazi angakhokelela ekuhlaselweni kwentliziyo kunye nokubetha. E-United States, i-ticagrelor yaqala ukuvunywa yi-FDA ngoJulayi 2011 yonyango lwezigulane zabantu abadala abane-acute coronary syndrome (ACS). Idatha yeklinikhi ibonisa ukuba i-ticagrelor iphumelele kakhulu kune-clopidogrel ekunciphiseni ukufa kwe-cardiovascular kufa ubuncinane kwiinyanga ze-12 emva kwesiganeko se-ACS. Ukongezelela, i-ticagrelorChemicalbook iphinde yanciphisa iziganeko ze-stent thrombosis (ST) kwizigulane ezifumene i-stents ukunyanga i-ACS. NgoJuni 2020, i-AstraZeneca yabhengeza ukuba i-US Food and Drug Administration (FDA) ivume i-anticoagulant Brilinta (ticagrelor) ukuba isetyenziswe kwizigulana ezinengozi ephezulu ye-coronary artery disease (CAD) ukunciphisa umngcipheko wokuhlaselwa yintliziyo yokuqala. okanye umngcipheko wokuhlaselwa sistrowuku. NgoNovemba 2020, i-AstraZeneca yazisa ukuba i-US Food and Drug Administration (FDA) ivume isalathisi esitsha se-anticoagulant Brilinta (ticagrelor), ngokudibanisa ne-aspirin, kunyango lwe-ischemia enzima. Kwizigulane ezine-hemorrhagic stroke okanye i-high-risk transient ischemic attack (TIA), iyanciphisa umngcipheko we-stroke elandelayo.
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Umgubo: ingxowa yefoyile ephindwe kabini yealuminiyam yesampulu eyi-1kg, kunye ne-25kgs ngegubu ngalinye ngobuninzi
Ulwelo: ibhotile etywiniweyo kwisampulu ye-1L, kunye ne-25kgs ngegubu ngalinye ngobuninzi