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Litheko tse tobileng tsa fektheri Pregabalin CAS 148553-50-8 e nang le boleng bo holimo le theko e tlase ka ho fetisisa setokong se bolokehileng le se potlakileng sa pharmaceutical mahareng.

Lebitso la sehlahisoa: Pregabalin
Nomoro ea CAS: 148553-50-8
Foromo ea molek'hule: C8H17NO2
Boima ba 'mele: 159.23
Nomoro ea EINECS: 604-639-1

 

 

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    tlhahiso ea lihlahisoa

    Lebitso la sehlahisoa Pregabalin
    Nomoro ea CAS. 148553-50-8
    EINECS No. 159.23
    Botenya 1.0±0.1 g/cm3
    Ntho e belang 274.0±23.0 °C(E boletsoeng esale pele)
    Sebaka se qhibilihang 194-196°C
    flash point 9℃
    Mokhoa oa limolek'hule C8H17NO2
    Boima ba molek'hule 159.23
    Ponahalo Mokelikeli o se nang Mebala
    Maemo a polokelo 2-8°C

    video ea sehlahisoa

    Tlhaloso ea Sehlahisoa:

    Pregabalin ke meriana e oelang tlas'a sehlopha sa lithethefatsi tsa anticonvulsant. Pregabalin e tsoa ho gamma-aminobutyric acid (GABA), neurotransmitter tsamaisong ea methapo e bohareng. Ka mokhoa o hlophisitsoeng, e amana le GABA ea "neurotransmitter" ea inhibitory, empa mokhoa oa eona oa ts'ebetso o fapane. Mabapi le thepa ea 'mele, pregabalin ke kristale e tšoeu e tiileng. Litšobotsi tsa eona tsa ho qhibiliha li kenyelletsa ho se qhibidihe ka metsing le ho qhibidiha ka bolokolohi dihlaoloseng tsa polar organic. Pregabalin e fumaneha ka mefuta ea litekanyetso tsa molomo, joalo ka li-capsules kapa matlapa, bakeng sa tšebeliso ea bongaka.
    Pregabalin e sebelisoa hangata ho phekola maemo a fapaneng a bongaka, ho kenyelletsa bohloko ba neuropathic, fibromyalgia, le mefuta e meng ea ho tsietsana. E fana ka liphello tsa eona tsa phekolo ka ho tlama ho subunit ea alpha-2-delta ea liteishene tsa calcium tse nang le voltage-gated tsamaisong ea methapo e bohareng. Tlamahano ena e hlophisa phallo ea li-ion tsa calcium, e fokotsa ho lokolloa ha li-neurotransmitters, 'me ka hona e fokotsa thabo ea lisele tsa methapo.

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