CAS 1451-83-8 China e babatsehang moetsi oa thepa ka kotloloho thekiso e phahameng Quality Fast Delivery high costomers khotsofalo Ho tsamaisa thepa ka thepa e nepahetseng theko e nepahetseng High Purity
Tlhaloso ea Sehlahisoa
Pregabalin (Lyrica), e tsoang ho GABA e amanang haufi-ufi le gabapentin, e 'nile ea etsoa lipatlisiso tse pharaletseng bakeng sa katleho ea eona ea ho phekola maemo a kang generalized depression disorder (GAD), fibromyalgia, bohloko ba neuropathic, le ho tsieleha ha karolo e itseng. Ho bonahala e na le phello e lebisitsoeng ho feta a2-δ subunit ea likanale tsa calcium bokong ha e bapisoa le gabapentin. Pregabalin e ile ea fuoa tumello ea FDA qetellong ea 2004 bakeng sa phekolo ea bohloko ba neuropathic le lefu la sethoathoa. Ka 2008, e ile ea e-ba meriana ea pele e amohelehang bakeng sa tsamaiso ea fibromyalgia. Leha pregabalin e ile ea amoheloa bakeng sa kalafo ea GAD ho European Union ka 2006, ha e so fumane tumello ea FDA bakeng sa GAD United States ho tloha nakong ea ho ngola.
video ea sehlahisoa
Sesebelisoa sa Sehlahisoa
S-Enantiomer ea Pregabalin. Analogue ea GABA e sebelisoang joalo ka anticonvulsant. Anxiolytic analgesic e sebelisetsoang ho phekola bohloko ba peripheral neuropathic le fibromyalgia.
Pregabalin ke sethethefatsi sa anticonvulsant se sebelisetsoang mahlaba a neuropathic, e le pheko e thusang bakeng sa ho tsietsana ka mokhoa o itseng,generalized khatello ea maikutlo. E entsoe e le mohlahlami ea matla ho feta oa gabapentin. Pregabalin e rekisoa ke Pfizer tlasa lebitso la khoebo
tlhahiso ea lihlahisoa
Lebitso le Tloaelehileng | Pregabalin |
Nomoro ea CAS | 148553-50-8 |
Botenya | 1.0±0.1 g/cm3 |
Ntlha e belang | 274.0±23.0 °C ho 760 mmHg |
Foromo ea limolek'hule | C8H17NO2 |
Boima ba Molek'hule | 159.226 |
PSA | 63.32000 |
LogP | 1.12 |
EINECS | 604-639-1 |
Khatello ea Mouoane | 0.0±1.2 mmHg ho 25°C |
Index ea Refraction | 1.465 |