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Dihexa CAS 1401708-83-5 Warshada Shiinaha iibka tooska ah ee dhoofinta Badbaadada aad u fiican Tayada qaaliga ah ee qiimaha sarreeya

Dihexa (magaca koodhka horumarinta PNB-0408), oo sidoo kale loo yaqaan N-hexanoic-Tyr-Ile- (6) aminohexanoic amide, waa daawada oligopeptide ee laga soo qaatay angiotensin IV taas oo ku xidhan dareen sare oo ku saabsan koritaanka hepatocyte factor (HGF) waxayna xoojinaysaa firfircoonida soo dhaweeyaheeda, c-Met.

 

 

 

    Sharaxaada Alaabta

    La kulmay Xarunta ayaa la ogaaday inay si xoog leh u wanaajiso shaqada garashada ee moodooyinka xayawaanka ee cudurka Alzheimers-sida naafanimada maskaxda. Marka la eego dhaqdhaqaaqa neurotrophic, Dihexa waxaa la ogaaday inuu yahay toddoba amar oo ka xoog badan qodobka neurotrophic ee maskaxda ka soo jeeda.

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    Codsiga Alaabta

    N-Hexanoic-Try-Ile-(6)-amino Hexanoic amide (Dihexa) waa angiotensin IV analoog ahaan sida wakiilka ogaanshaha/antidementia.
    Dihexa, oo ah daawada oligopeptide, waa angiotensin IV angiotensin IV analog ah oo afka ka shaqaynaysa iyo maskaxda-maskaxda. Dihexa waxay ku xidhan tahay factor kobaca hepatocyte (HGF) oo leh xidhiidh sare (Kd=65 pM) waxayna xoojisaa waxqabadkeeda soo-dhoweeyaha, c-Met. Dihexa waxa ay soo bandhigtaa firfircoonida lidka ku ah waallida oo aad u fiican waxayna wanaajisaa shaqada garashada ee moodooyinka xayawaanka. Dihexa waxa laga yaabaa inay leedahay awood daawayn oo ah daawaynta cudurka Alzheimers.

    qeexitaanka alaabta

    Magaca Guud Dihexa
    Lambarka CAS 1401708-83-5
    Cufnaanta  
    1.1±0.1 g/cm3
    Barta karkaraya  
    866.2± 65.0 °C at 760 mmHg
    Qaanuunka molecular
    C27H44N4O5
    Miisaanka Molecular 504.662
    LogP  
    2.78
    EINECS
    227-005-2
    Cadaadis uumiga  
    0.0±0.3 mmHg at 25°C
    Tusmada Milicsiga
    1.529

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