Fekitari yakananga kutengesa Pregabalin CAS 148553-50-8 ine yakanakisa mhando uye yakaderera mutengo muzvitoro zvakachengeteka uye nekukurumidza kuendesa mishonga yepakati.
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Product name | Pregabalin |
CAS Nha. | 148553-50-8 |
EINECS Nha. | 159.23 |
Density | 1.0±0.1 g/cm3 |
Boiling point | 274.0±23.0 °C(Zvakafanotaurwa) |
Melting point | 194-196°C |
Flash point | 9℃ |
Molecular formula | C8H17NO2 |
Molecular uremu | 159.23 |
Chitarisiko | Colorless Liquid |
Kuchengetedza mamiriro | 2-8°C |
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Product Description:
Pregabalin mushonga unowira pasi pekirasi ye anticonvulsant zvinodhaka. Pregabalin inotorwa kubva ku gamma-aminobutyric acid (GABA), neurotransmitter iri pakati penheyo system. Zvimiro, inobatana neiyo inhibitory neurotransmitter GABA, asi maitiro ayo ekuita akasiyana. Panyaya yezvimiro zvemuviri, pregabalin ichena crystalline yakasimba. Kunyungudika kwayo kunosanganisira kusanyungudika mumvura uye kunyungudika zvakasununguka mu polar organic solvents. Pregabalin inowanikwa mumuromo dosage mafomu, senge capsules kana mahwendefa, ekushandiswa kwemishonga.
Pregabalin inowanzoshandiswa kurapa zvirwere zvakasiyana-siyana, kusanganisira neuropathic pain, fibromyalgia, uye mamwe marudzi ekugumburwa. Inoshandisa maitiro ayo ekurapa nekusunga kune alpha-2-delta subunit yevoltage-gated calcium channels mukati mehutano hwehutano. Kusunga uku kunogadzirisa kuwanda kwecalcium ions, kuderedza kuburitswa kwemaurotransmitters, uye nekudaro kudzikisa kunakidzwa kwemasero etsinga.
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