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CAS 1451-83-8 Saina fa'atosina lelei le fa'atau tu'usa'o maualuga Tulaga Anapogi Fa'aolaina maualuga maualuga le fa'amalieina Saogalemu fe'avea'i tau talafeagai Maualuga Maualuga

Na fa'afaigaluegaina e avea o se mea fa'atauva'a taua mo meafaitino mo le fa'aogaina o meaola, fa'ato'aga fa'ato'aga, vaila'au ma vaila'au.

    Fa'amatalaga o oloa

    O le Pregabalin (Lyrica), o se mea e maua mai i le GABA e fesoʻotaʻi vavalalata ma le gabapentin, ua faia suʻesuʻega tele mo lona aoga i le togafitia o tulaga e pei o le faʻalavelave popole lautele (GAD), fibromyalgia, tiga o le neuropathic, ma vaega faʻalavelave faʻalavelave. E foliga mai o loʻo i ai se aʻafiaga sili atu i luga ole a2-δ subunit o ala calcium ile faiʻai pe a faʻatusatusa ile gabapentin. Pregabalin na tuʻuina atu le faʻamaoniga a le FDA i le faaiuga o le 2004 mo togafitiga o tiga o le neuropathic ma epilepsy. I le 2008, na avea ma vailaʻau muamua na faʻamaonia mo le puleaina o le fibromyalgia. E ui na faʻamaonia le pregabalin mo togafitiga GAD i le Europa Europa i le 2006, e leʻi mauaina le faʻamaoniga a le FDA mo GAD i le Iunaite Setete e pei o le taimi o le tusitusi.

    vitio oloa

    Talosaga Oloa

    S-Enantiomer o Pregabalin. O se GABA analogue faʻaaogaina e fai ma anticonvulsant. Anxiolytic analgesic faʻaaogaina e togafitia ai tiga neuropathic peripheral ma fibromyalgia.
    O le Pregabalin o se vailaʻau faʻamaʻi e faʻaaogaina mo tiga o le neuropathic, e fai ma togafitiga faʻaopoopo mo vaega faoa faamalosi, ma i totonu.lautele faaletonu popole. Na mamanuina e avea o se sui sili atu ona malosi i le gabapentin. Pregabalin o loʻo maketiina e Pfizer i lalo o le igoa tau fefaʻatauaʻiga

    fa'amatalaga o oloa

    Igoa masani Pregabalin
    Numera CAS 148553-50-8
    Malosi  
    1.0±0.1 g/cm3
    Fa'apuna  
    274.0±23.0 °C ile 760 mmHg
    Fuafua mole
    C8H17NO2
    Molecular Weight 159.226
    PSA  
    63.32000
    LogP  
    1.12
    EINECS
    604-639-1
    Omiga ausa  
    0.0±1.2 mmHg ile 25°C
    Fa'asinoga o le Fa'afoliga
    1.465

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