Uruganda rutanga ibikoresho bito CAS 863288-34-0 CJC-1295 (Nta DAC) Ifu ihamye Kugura kubakiriya Umutekano wohereza ibicuruzwa bishyushye bigurishwa
Gukoresha ibicuruzwa
Kurwanya gusaza: CJC1295 ikoreshwa murwego rwo kurwanya gusaza kugirango itume imisemburo ikura irekurwa. Uburyo bwibikorwa byabwo bukubiyemo guhuza reseptor zihariye muri glande ya pitoito, biganisha ku gusohora imisemburo ikura. Ibi birashobora gufasha guteza imbere gusana ingirabuzimafatizo, kongera imitsi, no kuzamura ubuzima muri rusange.
ibicuruzwa
URUBANZA No. | 863288-34-0 |
Inzira | C35H48N10O15 |
Uburemere bwa molekile | 3367.897 |
Ubucucike | 1.4 ± 0.1 g / cm3 |
Misa nyayo | 3365.893555 |
PSA | 1513.38000 |
LogP | -2.88 |
Ironderero | 1.644 |
Ibisobanuro ku bicuruzwa
CJC1295 ni imiti ivanze na CAS nimero 863288-34-0. Ni peptide ya sintetike igizwe nicyiciro cyimisemburo ikura ya hormone irekura (GHRH). CJC1295 igaragara nkifu yera idafite impumuro itandukanye. Imiterere yibanze igizwe numurongo wa aside amine. Inzira ya molekuline ya CJC1295 ni C165H269N47O46. Uru ruganda rushobora gushonga mumazi. Amakuru yumutekano yerekeye CJC1295 ntabwo aboneka muriki gihe. Ubundi bushakashatsi burakenewe kugirango umenye imiterere yumutekano.
Imirima ikoreshwa
Kurwanya gusaza: CJC1295 ikoreshwa murwego rwo kurwanya gusaza kugirango itume imisemburo ikura irekurwa. Uburyo bwibikorwa byabwo bukubiyemo guhuza reseptor zihariye muri glande ya pitoito, biganisha ku gusohora imisemburo ikura. Ibi birashobora gufasha guteza imbere gusana ingirabuzimafatizo, kongera imitsi, no kuzamura ubuzima muri rusange.
Gukura kw'imitsi: CJC1295 nayo ikoreshwa murwego rwo gukura kw'imitsi no kuzamura imikorere. Uburyo bwibikorwa byabwo bikubiyemo gushishikariza umusaruro wa insuline imeze nkikura rya 1 (IGF-1), igira uruhare runini mu mikurire no gusana. Ibi birashobora gutuma imitsi yiyongera, imbaraga, no gukira.
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