Uruganda rutanga ibikoresho bibisi CAS 113-79-1 Argipressin Ubwiza Bwiza Bwiza Buke Buke Bwihuse Gutanga Byihuse Gutanga Umutekano Kohereza Ubuziranenge Bukuru 99%
Gukoresha ibicuruzwa
Argipressine ihuza na arginine vasopressine reseptor V1 hamwe na Kd ya 1.31 nM muri A7r5 imbeba aortic yoroshye yimitsi.
ibicuruzwa
URUBANZA No. | 113-79-1 |
Inzira | C46H65N15O12S2 |
Uburemere bwa molekile | 1084.2316 |
Ubucucike | 1.6 ± 0.1 g / cm3 |
Ingingo ya Flash | 113 ℃ |
Misa nyayo | 1083.437866 |
PSA | 512.03000 |
LogP | -5.99 |
Kugaragara | ifu yera |
Ironderero | 1.724 |
Imiterere yo kubika | 2-8 ° C. |
Ibisobanuro ku bicuruzwa
ChEBI: Ubwoko bwiganje bwa vasopressine y’inyamabere (hormone antidiuretic). Ni nonapeptide irimo arginine isigaranye 8 na sisitemu ebyiri zifitanye isano na disulfide ku bisigisigi bya 1 na 6.Vasopressine tannate (PitressinTannate) ni tannate y'amazi adashobora gushonga ya vasopressine ikoreshwa mu buryo butemewe (ibice 1.5-5.0 by'ibinyamakuru buri munsi) igihe kirekire. Igikorwa nukurekura buhoro kwavasopressine.
Imirima ikoreshwa
Argipressine nuburyo bwiganje bwa vasopressine yinyamabere (hormone antidiuretic). Ni nonapeptide irimo arginine ku gisigara cya 8 na sisitemu ebyiri zifitanye isano na disulfide ku bisigisigi bya 1 na 6. Ifite uruhare nk'imiti y'umutima n'imitsi, imiti ivura indwara ya mitiweli na mitogen. | Ingaruka ya physiologique ya vasopressine ikoresheje Vasoconstriction. , na Kugabanuka kwa Diuresis. | Argipressin ni peptide ya syntetique ihwanye na hormone ya nonapeptide ya endogenous hamwe na antidiuretic. Gukomatanya muri hypothalamus no kubikwa / kurekurwa bivuye inyuma yinyuma ya pitoito, umurimo wibanze wa argipressin ni uguhuza ingano y’amazi adasanzwe. Iyi mikorere irashobora kandi gukora nka vasoconstrictor, ikongera umuvuduko wamaraso hamwe na sisitemu yo kurwanya imitsi. | Ubwoko bwiganjemo imisemburo ya antidiuretic yinyamabere. Ni nonapeptide irimo ARGININE ku gisigara cya 8 na sisitemu ebyiri zifitanye isano na disulfide ku bisigisigi bya 1 na 6. Arg-vasopressine ikoreshwa mu kuvura DIABETES INSIPIDUS cyangwa kunoza amajwi ya vasomotor hamwe n’AMARASO Y’AMARASO.
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