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Dihexa CAS 1401708-83-5 Uruganda rwo mu Bushinwa kugurisha mu buryo butaziguye Umutekano wohereza ibicuruzwa byiza Ubwiza buhebuje bw'abaguzi banyuzwe Kwihuta Gutanga byihuse Ibiciro Byera

Dihexa (izina ryizina ryiterambere PNB-0408), rizwi kandi nka N-hexanoic-Tyr-Ile- (6) aminohexanoic amide, ni umuti wa oligopeptide ukomoka kuri angiotensin IV uhuza cyane n’ikura rya hepatocyte (HGF) kandi ugatanga imbaraga zawo ibikorwa kuri reseptor yayo, c-Met.

 

 

 

    Ibisobanuro ku bicuruzwa

    Met. Urwo ruganda rwasanze rutezimbere cyane imikorere yubwenge mubyitegererezo byinyamanswa zindwara ya Alzheimer nkubumuga bwo mumutwe. Mu bushakashatsi bwakozwe ku bikorwa bya neurotrophique, Dihexa yasanze ari indwi ndwi z'ubunini zikomeye kuruta ubwonko bukomoka mu bwonko.

    videwo y'ibicuruzwa

    Gusaba ibicuruzwa

    N-Hexanoic-Gerageza-Ile- (6) -amino Hexanoic amide (Dihexa) nikigereranyo cya angiotensin IV nkumukozi wimenyekanisha / antidementia.
    Dihexa, imiti ya oligopeptide, ni umunwa ukora kandi mu maraso n'ubwonko-bwenge bwa angiotensin IV. Dihexa ihuza ibintu byo gukura kwa hepatocyte (HGF) hamwe cyane (Kd = 65 pM) kandi ikongerera imbaraga ibikorwa byayo kuri reseptor yayo, c-Met. Dihexa yerekana ibikorwa byiza byo kurwanya antidementia kandi itezimbere imikorere yubwenge mubyitegererezo byinyamaswa. Dihexa irashobora kugira ubushobozi bwo kuvura nkumuti wa Alzheimer.

    ibicuruzwa

    Izina Rusange Dihexa
    Umubare CAS 1401708-83-5
    Ubucucike  
    1.1 ± 0.1 g / cm3
    Ingingo  
    866.2 ± 65.0 ° C kuri 760 mmHg
    Inzira ya molekulari
    C27H44N4O5
    Uburemere bwa molekile 504.662
    LogP  
    2.78
    EINECS
    227-005-2
    Umuvuduko w'umwuka  
    0.0 ± 0.3 mmHg kuri 25 ° C.
    Ironderero ryo Kuvunika
    1.529

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