Manufacturer High Purity 98% Peptides Powder Liraglutide CAS 204656-20-2 Peptides Paura i roto i nga Vials iti utu iti peptides ataahua Paahua rawa mata
whakaritenga hua
ingoa hua | Liraglutide |
CAS No. | 204656-20-2 |
EINECS No. | 810-818-7 |
Kiato | N/A |
Kohuatanga | N/A |
Te rewa | N/A |
Ira hiko | N/A |
tātai rāpoi ngota | C172H265N43O51 |
Te taumaha ngota | 3751.202 |
Te ahua | Paura ma |
Nga tikanga rokiroki | -20°C |
ataata hua
Whakaahuatanga Hua
Ko te Liraglutide (NN2211) he glucagon-rite peptide-1 agonist-agonist-a-roa. I hokona i raro i te ingoa waitohu Victoza, he rongoa werohanga i hangaia e Novo Nordisk mo te maimoatanga o te mate huka momo 2. I te tau 2015, i timata a Novo Nordisk ki te hokohoko i te US i raro i te ingoa tohu liraglutide hei maimoatanga mo te momi i roto i nga pakeke me te iti rawa o te mate taumaha e pa ana ki te taumaha.
Nga Whakamahinga Hauora
Ko te Liraglutide he huanga werohanga kotahi ia ra o te incretin tangata (metabolic hormone) glucagon-like peptide-1 (GLP-1), mo te maimoatanga o te mate huka momo 2 me te momi.
Momo mate huka 2
Ko te Liraglutide te whakapai ake i te whakahaere o te huka toto. Te whakaroa i te puhanga o te kopu, me te pehi i te hunanga o te glucagon prandial.
He rite tonu ki nga tohu rereke me etahi atu agonists kaikawe GLP-1, he pai ake te liraglutide ki nga rongoa tuku iho mo te mate huka momo 2:
Kei a ia te kaha mo te aukati i te apoptosis me te whakaongaonga i te whakaoranga o nga pūtau beta (ka kitea i roto i nga rangahau kararehe).
Ka whakahekehia te hiahia me te aukati i te piki o te taumaha o te tinana, penei i te rangahau mahunga ki te upoko ki te glimepiride.
Ka whakahekehia nga taumata triglyceride toto.
Te momona
Kua whakaaetia a Liraglutide hei taapiri whakauru ki te kai iti-calorie me te whakanui ake i te korikori tinana mo te whakahaere taumaha i nga turoro pakeke. Ko nga paearu kua tohua ko te taurangi papatipu tinana tuatahi (BMI) o te 30 kg/m2 nui ake ranei (momomomo), 27 kg/m2 nui ake ranei (te taumaha rawa), i te mea ka pa mai te mate kino e pa ana ki te taumaha (hei tauira, te whakaheke toto, mate huka momo 2, dyslipidemia ranei). I te mutunga o te tau 2014, i purongohia nga raraunga mai i te whakamatautau SCALE™ Obesity and Prediabetes, he whakamatautau matapōkere, matarua-rua, e whakahaerehia ana e te placebo, he whakamatautau mo nga iwi maha i roto i te hunga kore-mate huka me te hunga momaa me te hunga kore-mate huka e taumaha ana ki nga mate comorbidities. I roto i tenei waahanga 3a whakamatautau, he 3,731 nga kaiuru kua tohatohahia ki te maimoatanga me te liraglutide 3 mg me te placebo ranei, e rua me te kai me te mahi. Ko te hunga i whakaoti i te whakamatautau 56-wiki i tutuki i te mate taimaha toharite o te 9.2%, kia whakaritea ki te 3.5% te whakaheke i te roopu placebo.
wa arahi
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