CAS 1451-83-8 Haina tino pai te kaihanga hoko tika te kounga teitei Ko te tuku tere te utu utu nui te pai o te utu kaipuke utu tika Te parakore teitei
Whakaahuatanga Hua
Ko te Pregabalin (Lyrica), he whakaputanga o te GABA e hono tata ana ki te gabapentin, kua rangahauhia e ia mo tona kaha ki te rongoa i nga ahuatanga penei i te mate awangawanga whanui (GAD), te fibromyalgia, te mamae neuropathic, me nga hopukanga matatini. Ko te ahua he nui ake te paanga ki te waahanga a2-δ o nga awa konupūmā i roto i te roro ka whakaritea ki te gabapentin. I whakawhiwhia a Pregabalin i te whakaaetanga FDA i te mutunga o te 2004 mo te maimoatanga o te mamae neuropathic me te epilepsy. I te 2008, ko te rongoa tuatahi i whakaaetia mo te whakahaere o te fibromyalgia. Ahakoa i whakaaetia te pregabalin mo te maimoatanga GAD i te Kotahitanga o Europi i te tau 2006, kaore ano kia whiwhi whakaaetanga FDA mo GAD i te United States i te wa o te tuhi.
ataata hua
Tono Hua
S-Enantiomer o Pregabalin. He riterite GABA i whakamahia hei anticonvulsant. Anxiolytic analgesic whakamahia ki te hamani mamae neuropathic peripheral me te fibromyalgia.
Ko te Pregabalin he rongoa anticonvulsant e whakamahia ana mo te mamae neuropathic, hei rongoa taapiri mo te hopu i etahi waahanga, me tewhānui raruraru ohorere. I hangaia hei whakakapi kaha ake ki te gabapentin. Kei te maakete a Pregabalin e Pfizer i raro i te ingoa hokohoko
whakaritenga hua
Ingoa noa | Pregabalin |
Tau CAS | 148553-50-8 |
Kiato | 1.0±0.1 g/cm3 |
Kohuatanga | 274.0±23.0 °C i te 760 mmHg |
Tātai rāpoi | C8H17NO2 |
Taumaha rāpoi | 159.226 |
PSA | 63.32000 |
RangitakiP | 1.12 |
EINECS | 604-639-1 |
Pehenga Kohu | 0.0±1.2 mmHg i te 25°C |
Taurangi o te Refraction | 1.465 |