Ahịa ụlọ ọrụ Pregabalin CAS 148553-50-8 nwere ezigbo mma yana ọnụ ala dị ala na ngwaahịa nchekwa na nnyefe ngwa ngwa ọgwụ etiti.
nkọwapụta ngwaahịa
Aha ngwaahịa | Pregabalin |
CAS Mba. | 148553-50-8 |
EINECS Mba. | 159.23 |
Njupụta | 1.0±0.1 g/cm3 |
Ebe esi nri | 274.0± 23.0 Celsius C (buru amụma) |
Ebe mgbaze | 194-196°C |
ebe mgbari | 9 ℃ |
Usoro ihe omimi | C8H17NO2 |
Ibu molekụla | 159.23 |
Ọdịdị | Mmiri na-enweghị agba |
Ọnọdụ nchekwa | 2-8 Celsius C |
vidiyo ngwaahịa
Nkọwa ngwaahịa:
Pregabalin bụ ọgwụ na-adaba n'okpuru klas nke ọgwụ mgbochi mkpali. Pregabalin bụ ihe sitere na gamma-aminobutyric acid (GABA), onye na-ebugharị neurotransmitter na sistemu ụjọ nke etiti. N'usoro, ọ metụtara GABA neurotransmitter inhibitory, mana usoro ya dị iche. N'ihe gbasara akụrụngwa anụ ahụ, pregabalin bụ kristal ọcha siri ike. Njirimara solubility ya na-agụnye ịbụ ihe a na-adịghị ahụkebe na mmiri yana soluble kpamkpam n'ime ihe ndị na-agbaze organic pola. Pregabalin dị n'ụdị usoro onunu, dị ka capsules ma ọ bụ mbadamba, maka iji ọgwụ.
A na-ejikarị Pregabalin na-agwọ ọnọdụ ahụike dị iche iche, gụnyere mgbu neuropathic, fibromyalgia, na ụfọdụ ụdị ọdịdọ. Ọ na-egosipụta mmetụta ọgwụgwọ ya site na ijikọ na mpaghara alfa-2-delta nke chanel calcium voltaji na sistemụ ụjọ etiti. Nke a na-ejikọta ọnụ na-agbanwe mbata nke calcium ion, na-ebelata ntọhapụ nke neurotransmitters, ma si otú ahụ na-ebelata mkpali nke mkpụrụ ndụ akwara.
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