Na-ere ọkụ na-ere CAS 52232-67-4 Teriparatide acetate ezigbo ọnụahịa nchekwa nnyefe dị elu ngwaahịa ire ere ọkụ na afọ ojuju ndị ahịa dị elu.
nkọwapụta ngwaahịa
Aha nkịtị | Teriparatide acetate |
Nọmba CAS | 52232-67-4 |
Ibu molekụla | 4177.77000 |
Usoro ihe omimi | C181H291N55O51S2 |
EINECS | 640-978-1 |
Nkwụsi ike | Hygroscopic |
Ọdịdị | ntụ ntụ |
Ọnọdụ nchekwa | -20°C |
Video ngwaahịa
Eji ngwaahịa
Teriparatide bụ agonist nke PHT, na uru IC50 dị na sel HEK293 bụ 2 nM.Teripartite nwere ike ime ka ọkpụkpụ na-edozi ahụ site na igbochi osteoblast apoptosis, na-eme ka ọkpụkpụ ọkpụkpụ na-eme ka ọkpụkpụ ọkpụkpụ na-eme ka ọdịiche dị iche iche nke osteoblast dịkwuo mma. Site n'ịchịkwa adenylate cyclase-cyclic adenosine monophosphate-protein kinase A ụzọ, PHT-ⅰ anabata n'elu osteoblasts, ọkpụkpụ lining cell na ụmị ọkpụkpụ stromal sel na-akpalite intermittently iji kwalite ọdịiche nke osteoblasts na ogologo ndụ ha. Na-akpali mmụba nke ahịrị sel osteobast site na phosphate C- cytoplasmic calcium ion-protein kinase Chemibook C ụzọ ntụgharị akara; Site na igbochi ọrụ trans-activation nke PPARγ, ọdịiche nke mkpụrụ ndụ stromal n'ime ahịrị adipocyte na-ebelata na ọnụ ọgụgụ osteoblasts na-abawanye. Ụkpụrụ na-apụtaghị ìhè nke uto ọkpụkpụ site n'ịchịkwa cytokines, dịka ọmụmaatụ, nwere ike ime ka iGF-1 jikọta ya na osteoblasts, si otú ahụ na-akwalite ọkpụkpụ ọkpụkpụ; Ụzọ akara Wnt na-achịkwa usoro nhazi ọkpụkpụ, si otú a na-amụba ọkpụkpụ ọkpụkpụ.
Ozi ụlọ ọrụ
Demei Pharmaceutical Technology Co., Ltd. bụ ụlọ ọrụ siri ike na nke ọhụrụ ọkachamara na nyocha, nrụpụta na nkesa nke ngwa ọgwụ dị elu na ogige organic. Site na ntinye siri ike iji kwalite ụlọ ọrụ ọgwụ zuru ụwa ọnụ, anyị na-arara onwe anyị nye ikwado mbupụ nke ngwaahịa ọgwụ ndị China n'ụwa niile. Pọtụfoliyo ngwaahịa anyị buru ibu enwetala amara n'ahịa ndị bụ isi, gụnyere UK, Germany, Australia, Netherlands, Poland, Russia, Kazakhstan, Philippines, Malaysia, Singapore na ọtụtụ mpaghara ndị ọzọ. N'ịnabata ụkpụrụ nke iguzosi ike n'ezi ihe na nghọta, anyị na-ebute ụzọ iwulite mmekọrịta ntụkwasị obi na ndị ahịa anyị, na-ahụ na ọganiihu n'otu n'otu na mmekọrịta dị ogologo oge.
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