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CAS 1451-83-8 China magburu onwe ya nrụpụta ụlọ ahịa na-ere ahịa dị elu Ogo Nnyefe ngwa ngwa dị elu ndị ahịa afọ ojuju Mbupu nchekwa kwesịrị ekwesị ọnụahịa dị ọcha

Ọ rụrụ ọrụ dị ka ihe dị mkpa etiti maka akụrụngwa maka organic njikọ, agrochemical, ọgwụ na dyestuff ubi.

    Nkọwa ngwaahịa

    Pregabalin (Lyrica), ihe sitere na GABA nke nwere njikọ chiri anya na gabapentin, emeela nyocha dị ukwuu maka ịdị irè ya n'ịgwọ ọnọdụ ndị dị ka nsogbu nchekasị zuru oke (GAD), fibromyalgia, mgbu neuropathic, na nkwụsịtụ mgbagwoju anya. Ọ dị ka ọ nwere mmetụta ezubere iche karịa na mpaghara a2-δ nke ọwa calcium na ụbụrụ ma e jiri ya tụnyere gabapentin. Enyere Pregabalin nkwado FDA na njedebe nke 2004 maka ọgwụgwọ nke mgbu neuropathic na akwụkwụ. Na 2008, ọ ghọrọ ọgwụ mbụ akwadoro maka njikwa fibromyalgia. Ọ bụ ezie na a kwadoro pregabalin maka ọgwụgwọ GAD na European Union na 2006, ọ nwetabeghị nkwado FDA maka GAD na United States dị ka n'oge ederede.

    vidiyo ngwaahịa

    Ngwa ngwaahịa

    S-Enantiomer nke Pregabalin. Analọgụ GABA ejiri dị ka ọgwụ mgbochi. Anxiolytic analgesic na-eji na-emeso mgbu neuropathic mpụta na fibromyalgia.
    Pregabalin bụ ọgwụ anticonvulsant ejiri mee ihe maka mgbu neuropathic, dị ka ọgwụgwọ mgbakwunye maka ọdịdọ akụkụ, yanamkpokọta nsogbu nchekasị. Emebere ya ka ọ bụrụ onye ga-anọchi gabapentin karịa. Pfizer na-ere Pregabalin n'okpuru aha ahia

    nkọwapụta ngwaahịa

    Aha nkịtị Pregabalin
    Nọmba CAS 148553-50-8
    Njupụta  
    1.0±0.1 g/cm3
    Ebe esi nri  
    274.0± 23.0 °C na 760 mmHg
    Usoro ihe omimi
    C8H17NO2
    Ibu molekụla 159.226
    PSA  
    63.32000
    LogP  
    1.12
    EINECS
    604-639-1
    Uzuoku Nrụgide  
    0.0±1.2 mmHg na 25°C
    Index nke ntụgharị uche
    1.465

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