Stable Buyback daga Abokan ciniki CAS 16789-98-3 Desmopressin Maƙerin Maƙeran Ma'adinan Halitta Mai Kaya Mai Tsabtataccen Tsafta 99%
Amfani da samfur
Desmopressin acetate (DDAVP, Micondensate), wanda shine deamination na 1-cysteine da maye gurbin 8-L-arginine tare da 8-D-arginine, wanda kuma aka sani da aminoarginine vasopressin, shine tsarin tsarin analog na halitta arginine gishiri vasopressin da abin da aka samo asali. da vasopressin. Its antidiuretic sakamako ne mafi ƙarfi da dawwama fiye da na vasopressin, amma ba shi da wani vasoconstriction sakamako kuma yana da 'yan illa. An yi amfani da shi a asibiti ta hanyar asibiti ko rashin aikin platelet, uremia, cirrhosis na hanta da kuma tsawon lokacin zubar jini wanda ba a sani ba; za a iya amfani dashi don sarrafawa da hana zubar jini a lokacin ƙananan tiyata; tsakiyar ciwon sukari insipidus, da dai sauransu. A cikin mutum lokuta, wannan samfurin na iya ma zama tasiri a marasa lafiya da matsakaici urinary tsarin cuta, kuma sau da yawa contraindicated a marasa lafiya da irin IIB von Willebrand cuta.
ƙayyadaddun samfur
CAS No. | 16789-98-3 |
Formula | Saukewa: C186H286N50O62S |
Yawan yawa | 1.56 g/cm 3 |
Nauyin kwayoyin halitta | 1129.269 |
Daidai taro | 1128.448120 |
PSA | 560.61000 |
LogP | 1.70530 |
Yanayin ajiya | an rufe kuma an kiyaye shi daga haske |
Bayanin samfur
Desmopressin acetate (DDAVP, Stimate) shine roba 1-desamino-8-D-argininevasopressin. Ingancin sa, sauƙin gudanarwa (intranasal), tsawon lokacin aiki, da rashin sakamako masu illa sun sa shi zaɓin zaɓi don kula da ciwon sukari na tsakiya. Hakanan za'a iya gudanar da shi ta hanyar intramuscularly ta hanyar travenously. An fi son yin allurar vasopressin da maganin antidiuretics na baki don amfani a cikin yara. An nuna shi gudanar da polydipsia na wucin gadi da polyurias wanda ke da alaƙa da rauni zuwa
Analog na roba na hormone pituitary, ARGININE VASOPRESSIN. Ayyukansa yana yin sulhu ta hanyar mai karɓar VASOPRESSIN V2. Yana da aikin antidiuretic na tsawon lokaci, amma ƙananan tasirin latsawa. Hakanan yana daidaita matakan kewayawa FACTOR VIII da VON WILLEBRAND FACTOR.
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