Kasuwancin masana'antu kai tsaye Pregabalin CAS 148553-50-8 tare da mafi kyawun inganci da mafi ƙarancin farashi a cikin aminci da isar da sauri na magunguna na tsakiya
ƙayyadaddun samfur
Sunan samfur | Pregabalin |
CAS No. | 148553-50-8 |
EINECS No. | 159.23 |
Yawan yawa | 1.0± 0.1 g/cm3 |
Wurin tafasa | 274.0 ± 23.0 °C (An annabta) |
Wurin narkewa | 194-196 ° C |
Wurin walƙiya | 9 ℃ |
Tsarin kwayoyin halitta | Saukewa: C8H17NO2 |
Nauyin kwayoyin halitta | 159.23 |
Bayyanar | Ruwa mara launi |
Yanayin ajiya | 2-8 ° C |
samfurin bidiyo
Bayanin samfur:
Pregabalin magani ne da ke faɗuwa a ƙarƙashin ajin magungunan kashe-kashe. Pregabalin ya samo asali ne daga gamma-aminobutyric acid (GABA), mai watsawa a cikin tsarin juyayi na tsakiya. A tsari, yana da alaƙa da GABA neurotransmitter mai hanawa, amma tsarin aikinsa ya bambanta. Dangane da kaddarorin jiki, pregabalin wani farin kristal ne mai ƙarfi. Halayen solubility ɗin sa sun haɗa da kasancewa a zahiri ba a iya narkewa a cikin ruwa kuma ana iya narkewa cikin yardar rai a cikin kaushi na kwayoyin halitta. Ana samun Pregabalin a cikin nau'ikan sashi na baka, kamar capsules ko allunan, don amfanin magani.
Ana amfani da Pregabalin akai-akai don magance yanayin kiwon lafiya daban-daban, gami da ciwon neuropathic, fibromyalgia, da wasu nau'ikan rikice-rikice. Yana aiwatar da tasirinsa na warkewa ta hanyar ɗaure ga sashin alpha-2-delta na tashoshin calcium mai ƙarfin lantarki a cikin tsarin juyayi na tsakiya. Wannan ɗaure yana daidaita kwararar ions na calcium, yana rage sakin ƙwayoyin jijiya, kuma ta haka yana rage haɓakar ƙwayoyin jijiya.
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