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CAS 204656-20-2 Liraglutide China kyakkyawan masana'anta kai tsaye tallace-tallace Babban Tsafta Tsaro jigilar kaya mai inganci daidai farashin manyan masu siye gamsuwa da Isar da sauri

Liraglutide, lipopeptide da polypeptide, analog ne na ɗan adam GLP-1 wanda ragowar lysine a matsayi na 27 aka maye gurbinsa da arginine da ƙungiyar hexadecanoyl da aka haɗe zuwa ragowar lysine ta hanyar sararin samaniyar glutamic acid. Ana amfani dashi tare da abinci da motsa jiki don haɓaka sarrafa glycemic a cikin manya masu fama da ciwon sukari na 2. Liraglutide yana aiki azaman glucagon-kamar peptide-1 agonist mai karɓa kuma yana aiki azaman wakili na neuroprotective.

 

 

 

 

    Bayanin samfur

    Liraglutide shine GLP-1 (1-37) wanda aka gyara a Ly: ƙungiyar -amino an haɗa shi da wani nau'in (N-hexadecanoyl) glutam--yl wanda ba tare da haɗin gwiwa ba amma yana ɗaure ɗan adam albumin. (Har ila yau, an maye gurbin Lys tare da Arg.) Waɗannan canje-canje suna ba da damar ƙara yawan jini t1?2 na 10 zuwa 15 hours bayan gudanarwar sc (0.6-1.8 MG), yana ba da damar yin amfani da sau ɗaya kowace rana. Liraglutide (Victoza, Novo Nordisk) yana jiran amincewar FDA, EMEA, da Koˉ roˉ -shoˉ (Japan).

    samfurin bidiyo

    Aikace-aikacen samfur

    Liraglutide wani sabon nau'in maganin hypoglycemic ne wanda ke kunna furotin da ke kunna AMP don haka yana haɓaka hankalin insulin. Ba wai kawai yana da tasiri mai mahimmanci na hypoglycemic ba, har ma yana da ayyuka na asarar nauyi, rage karfin jini, da haɓaka bayanan lipid na jini.
    Liraglutide, ɗan adam glucagon-kamar peptide-1 (GLP-1) agonist mai karɓa, yana jinkirin zubar ciki, yana ƙara koshi, kuma yana rage cin abinci mara lafiya, yayin da rage sha'awar ci da ƙyale jiki don ƙara yawan kashe kuzari yana taka rawa wajen nauyi. hasara; yana hana hanta samar da glucose da yawa kuma yana inganta pancreas don samar da ƙarin insulin don rage sukarin jini; Bugu da kari, liraglutide kuma yana da fa'idodin zuciya da jijiyoyin jini da kuma kariyar koda.

    ƙayyadaddun samfur

    Sunan gama gari Liraglutide
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